Page 115 - 南京医科大学自然版
P. 115
第45卷第1期 谢 佺,周雨萱,蔡舒玥,等. 用于前列腺癌诊疗的PSMA 靶向放射性小分子探针研究进展[J].
2025年1月 南京医科大学学报(自然科学版),2025,45(1):105-110 ·109 ·
therapy for prostate cancer[J]. Prostate Cancer Prostatic 2015,56(6):914-920
Dis,2022,25(1):11-26 [20]WEINEISEN M,SIMECEK J,SCHOTTELIUS M,et al.
[9] FAROLFI A,CALDERONI L,MATTANA F,et al. Cur⁃ Synthesis and preclinical evaluation of DOTAGA⁃conju⁃
rent and emerging clinical applications of PSMA PET di⁃ gated PSMA ligands for functional imaging and endoradio⁃
agnostic imaging for prostate cancer[J]. J Nucl Med, therapy of prostate cancer[J]. EJNMMI Res,2014,4(1):
2021,62(5):596-604 63
[10]MOUL J W,SHORE N D,PIENTA K J,et al. Application [21]WEINEISEN M,SCHOTTELIUS M,SIMECEK J,et al.
of next ⁃ generation imaging in biochemically recurrent 68 Ga⁃ and 177 Lu⁃labeled PSMA I&T:optimization of a PS⁃
prostate cancer[J]. Prostate Cancer Prostatic Dis,2024, MA⁃targeted theranostic concept and first proof⁃of⁃con⁃
27(2):202-211 cept human studies[J]. J Nucl Med,2015,56(8):1169-
[11]许馨晨,顾莹莹,唐立钧. 影像组学在前列腺癌中的研 1176
68
究进展[J].南京医科大学学报(自然科学版),2024,44 [22]CYTAWA W,SEITZ A K,KIRCHER S,et al. Ga⁃PSMA
(7):1010-1017 I&T PET/CT for primary staging of prostate cancer[J].
XU C X,GU Y Y,TANG L J. Advances of radiomics in Eur J Nucl Med Mol Imaging,2020,47(1):168-177
prostate cancer[J]. Journal of Nanjing Medical University [23]EMMETT L,PAPA N,BUTEAU J,et al. The primary
68
(Nature Sciences),2024,44(7):1010-1017 score:using intraprostatic Ga⁃PSMA PET/CT patterns to
[12]JIAO J,ZHANG J,WEN W,et al. Prostate⁃specific mem⁃ optimize prostate cancer diagnosis[J]. J Nucl Med,2022,
brane antigen⁃targeted surgery in prostate cancer:accu⁃ 63(11):1644-1650
rate identification,real⁃time diagnosis,and precise resec⁃ [24]MEYER C,PRASAD V,STUPARU A,et al. Comparison
tion[J]. Theranostics,2024,14(7):2736-2756 of PSMA⁃TO⁃1 and PSMA⁃617 labeled with gallium⁃68,
[13]ELLS Z,GROGAN T R,CZERNIN J,et al. Dosimetry of lutetium⁃177 and actinium⁃225[J]. EJNMMI Res,2022,
177
[ Lu]Lu⁃PSMA⁃targeted radiopharmaceutical therapies 12(1):65
in patients with prostate cancer:a comparative systematic [25]LUNDMARK F,OLANDERS G,RINNE S S,et al. De⁃
review and metaanalysis[J]. J Nucl Med,2024,65(8): sign,synthesis,and evaluation of linker⁃optimised PSMA⁃
1264-1271 targeting radioligands[J]. Pharmaceutics,2022,14(5):
[14]SONG H,LEONIO M I,FERRI V,et al. Same⁃day post⁃ 1098
therapy imaging with a new generation whole⁃body digital [26]CHEN Y,ZHAN X,NI M,et al. Synthesis,preclinical
177
68
SPECT/CT in assessing treatment response to[ Lu]Lu⁃ evaluation,and first ⁃ in ⁃ human PET study of[ Ga]⁃ la⁃
PSMA⁃617 in metastatic castration⁃resistant prostate can⁃ beled biphenyl ⁃ containing PSMA tracers[J]. J Med
cer[J]. Eur J Nucl Med Mol Imaging,2024,51(9):2784- Chem,2023,66(18):13332-13345
68
2793 [27]DUAN X,CAO Z,ZHU H,et al. Ga⁃labeled ODAP⁃urea⁃
[15]CUI X Y,LI Z,KONG Z,et al. Covalent targeted radioli⁃ based PSMA agents in prostate cancer:first⁃in⁃human im⁃
gands potentiate radionuclide therapy[J]. Nature,2024, aging of an optimized agent[J]. Eur J Nucl Med Mol Imag⁃
630(8015):206-213 ing,2022,49(3):1030-1040
[16]JIA A Y,KIESS A P,LI Q,et al. Radiotheranostics in ad⁃ [28]HOU H,PAN Y,WANG Y,et al. Development and first⁃in⁃
vanced prostate cancer:current and future directions[J]. human study of PSMA ⁃ targeted PET tracers with im⁃
Prostate Cancer Prostatic Dis,2024,27(1):11-21 proved pharmacokinetic properties[J]. Eur J Nucl Med
68
[17]EDER M,SCHÄFER M,BAUDER⁃WÜST U,et al. Ga⁃ Mol Imaging,2024,51(9):2819-2832
complex lipophilicity and the targeting property of a urea⁃ [29]HOU H,LIN Y,PAN Y,et al. Synthesis and preclinical
68
based PSMA inhibitor for PET imaging[J]. Bioconjug evaluation of Ga ⁃ labeled PSMA tracers with improved
Chem,2012,23(4):688-697 pharmacological properties[J]. Eur J Med Chem,2024,
[18]SCHÄFER M,BAUDER⁃WÜST U,LEOTTA K,et al. A 274:116545
dimerizedurea⁃basedinhibitoroftheprostate⁃specificmem⁃ [30]MEASE R C,DUSICH C L,FOSS C A,et al. N⁃[N⁃[(S)⁃
18
68
brane antigen for Ga⁃PET imaging of prostate cancer[J]. 1,3⁃dicarboxypropyl]carbamoyl]⁃4⁃[ F]fluorobenzyl⁃L⁃
18
EJNMMI Res,2012,2(1):23 cysteine,[ F]DCFBC:a new imaging probe for prostate
[19]BENEŠOVÁ M,SCHÄFER M,BAUDER⁃WÜST U,et al. cancer[J]. Clin Cancer Res,2008,14(10):3036-3043
Preclinical evaluation of a tailor⁃made DOTA⁃conjugated [31]CHO S Y,GAGE K L,MRASE R C,et al. Biodistribution,
18
PSMA inhibitor with optimized linker moiety for imaging tumor detection,and radiation dosimetry of F⁃DCFBC,
and endoradiotherapy of prostate cancer[J]. J Nucl Med, a low ⁃ molecular ⁃ weight inhibitor of prostate ⁃ specific

